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8-Aryl-6-chloro-3-nitro-2-(phenylsulfonylmethyl)imidazo[1,2-a]pyridines as potent antitrypanosomatid molecules bioactivated by type 1 nitroreductases
Cyril Fersing
,
Clotilde Boudot
,
Julien Pedron
,
Sébastien Hutter
,
Nicolas Primas
,
et al.
Article dans une revue
hal-01909649v1
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8-Alkynyl-3-nitroimidazopyridines display potent antitrypanosomal activity against both T. b. brucei and cruzi
Cyril Fersing
,
Clotilde Boudot
,
Caroline Castera-Ducros
,
Émilie Pinault
,
Sébastien Hutter
,
et al.
Article dans une revue
hal-02899751v1
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6-Chloro-3-nitro-2-[(phenylsulfonyl)methyl]imidazo[1,2-b]pyridazine
Romain Paoli-Lombardo
,
Nicolas Primas
,
Sébastien Hutter
,
Sandra Bourgeade-Delmas
,
Clotilde Boudot
,
et al.
Article dans une revue
hal-04115477v1
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Novel 8-nitroquinolin-2(1 H )-ones as NTR-bioactivated antikinetoplastid molecules: Synthesis, electrochemical and SAR study
Julien Pedron
,
Clotilde Boudot
,
Sébastien Hutter
,
Sandra Bourgeade-Delmas
,
Jean-Luc Stigliani
,
et al.
Article dans une revue
hal-01888465v1
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Antikinetoplastid SAR study in 3-nitroimidazopyridine series
Cyril Fersing
,
Clotilde Boudot
,
Romain Paoli-Lombardo
,
Nicolas Primas
,
Emilie Pinault
,
et al.
Article dans une revue
hal-02920293v1
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Nongenotoxic 3-Nitroimidazo[1,2- a ]pyridines Are NTR1 Substrates That Display Potent in Vitro Antileishmanial Activity
Cyril Fersing
,
Louise Basmaciyan
,
Clotilde Boudot
,
Julien Pedron
,
Sébastien Hutter
,
et al.
Article dans une revue
hal-02478935v1
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Improving Aqueous Solubility and In Vitro Pharmacokinetic Properties of the 3-Nitroimidazo[1,2-a]pyridine Antileishmanial Pharmacophore
Romain Paoli-Lombardo
,
Nicolas Primas
,
Sandra Bourgeade-Delmas
,
Sébastien Hutter
,
Alix Sournia-Saquet
,
et al.
Article dans une revue
hal-03755519v1
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